255. "Diastereoselective Synthesis of Enantioenriched Trifluoromethylated Ethylenediamines and Isoindolines Containing Two Stereogenic Carbon Centers by Nucleophilic Trifluromethylation Using HFC-23"
Hirano, Kazuki; Saito Takuya; Fujihira, Yamato; Sedgwick, Daniel M.; Fustero, Santos; Shibata, Norio
J. Org. Chem. 2020, accepted for publication.
254. "The Ruthenium-Catalyzed Domino Cross Enyne Metathesis/Ring-Closing Metathesis in the Synthesis of Enantioenriched Nitrogen-Containing Heterocycles"
Alberto Llobat, Jorge Escorihuela, Daniel M. Sedgwick, Miriam Rodenes, Raquel Román, Vadim A. Soloshonok, Jianlin Han, Mercedes Medio-Simón, Santos Fustero.
Eur. J. Org. Chem. 2020, accepted for publication.
253. "Tailor-Made Amino Acids and Fluorinated Motifs as Prominent Traits in the Modern Pharmaceuticals"
Haibo Mei, Jianlin Han, Sarah White, Daniel J. Graham, Kunisuke Izawa, Tatsunori Sato, Santos Fustero, Nicholas A. Meanwell, Vadim A. Soloshonok
Chem. Eur. J. 2020, accepted for publication.
252. "Nucleic acid recognition and antiviral activity of 1,4-substituted terphenyl compounds mimicking all faces of the HIV1 Rev protein positively-charged α-helix"
Cristina Medina-Trillo, Daniel M. Sedgwick, Lidia Herrera, Manuela Beltrán, Ángela Moreno, Pablo Barrio, Luis M. Bedoya, José Alcamí, Santos Fustero, José Gallego
Scientific Reports (nature research) 2020, 10(1), 7190 (doi.org/10.1038/s41598-020-64120-2).
251. "Fluorine-containing drugs approved by the FDA in 2019"
Haibo Mei, Attila Márió Remete, Yupiao You, Hiroki Moriwaki, Santos Fustero, Lorand Kiss, Vadim Soloshonok, Jianlin Han
Chinese Chemistry Letters 2020, 31, early view.
250. "Asymmetric Synthesis of Fluorinated Monoterpenic Alkaloid Derivatives from Chiral Fluoroalkyl Aldimines via the Pauson-Khand Reaction"
Alberto Llobat, Daniel M. Sedgwick, Albert Cabré, Raquel Román, Natalia Mateu, Jorge Escorihuela, Mercedes Medio Simón, Vadim Soloshonok, Jianlin Han, Antoni Riera, Santos Fustero
Adv. Synth. Catal. 2020, 362, 1378-1384.